Histone Demethylase Inhibitors

KDM1/LSD1

KDM2

KDM3

KDM4

KDM5

KDM6

KDM7

Histone Demethylase Inhibitors, Antagonists, Degraders & Ligands

Product Name	KDM1/LSD1	KDM2	KDM3	KDM4	KDM5	KDM6	KDM7	Purity
GSK-J4						KDM6		99.45%
CPI-455					KDM5			98.95%
Tranylcypromine hydrochloride	LSD1							99.91%
TAS1440 benzoate	KDM1/LSD1, IC₅₀: 4.8 nM
IOX1		KDM2	KDM3	KDM4		KDM6		99.89%
GSK2879552	KDM1/LSD1							99.98%
JIB-04				KDM4	KDM5	KDM6		98.63%
Iadademstat dihydrochloride	KDM1/LSD1							99.98%
GSK-J4 hydrochloride						KDM6		99.01%
QC6352				KDM4A, IC₅₀: 104 nM KDM4B, IC₅₀: 56 nM KDM4C, IC₅₀: 35 nM KDM4D, IC₅₀: 104 nM	KDM5B, IC₅₀: 750 nM			99.13%
GSK-LSD1 dihydrochloride	KDM1/LSD1							99.88%
Iadademstat	LSD1							99.82%
KDM5-C70					KDM5			98.82%
GSK-J1						KDM6		99.94%
SP2509	KDM1/LSD1							99.50%
Tranylcypromine hemisulfate	KDM1/LSD1							99.94%
Daminozide		KDM2						99.79%
ML324				KDM4				98.35%
KDOAM-25 citrate					KDM5			98.56%
AS8351					KDM5			99.88%
GSK467					KDM5, Ki: 10 nM KDM5, IC₅₀: 26 nM			99.34%
Seclidemstat	KDM1/LSD1							99.77%
Pulrodemstat benzenesulfonate	KDM1/LSD1							99.64%
PFI-90			KDM3					99.86%
Zavondemstat				KDM4A, IC₅₀: ≤ 0.08 μM KDM4B, IC₅₀: ≤ 0.08 μM KDM4C, IC₅₀: ≤ 0.08 μM KDM4D, IC₅₀: ≤ 0.08 μM				99.29%
TK-129					KDM5, IC₅₀: 44 nM			≥98.0%
KDM2/7-IN-1		KDM2		KDM4			KDM7	99.9%
NCGC00244536				KDM4				99.70%
KDM5A-IN-1					KDM5			99.64%
Bomedemstat ditosylate	KDM1/LSD1							99.14%
KDM4C-IN-1				KDM4				98.13%
Bomedemstat	KDM1/LSD1							99.43%
TAK-418	KDM1/LSD1							99.81%
DDP-38003 dihydrochloride	KDM1/LSD1							99.31%
NSC636819				KDM4				98.90%
Bomedemstat hydrochloride	KDM1/LSD1							99.94%
CPI-455 hydrochloride					KDM5			99.95%
KDM2A/7A-IN-1		KDM2						99.94%
KDM5-IN-1					KDM5			99.52%
Seclidemstat mesylate	KDM1/LSD1							99.80%
JQKD82 trihydrochloride					KDM5			99.89%
KDM4D-IN-1				KDM4				98.82%
KDM2B-IN-4		KDM2						99.61%
LSD1/HDAC6-IN-2	LSD1, IC₅₀: 5 nM							99.66%
S2101	KDM1/LSD1							99.70%
T-448	KDM1/LSD1							98.86%
Bomedemstat dihydrochloride	KDM1/LSD1							99.55%
KDM4-IN-3				KDM4				99.36%
S234984	LSD1-CoREST							99.46%
Arborinine	LSD1							99.87%
PBIT					KDM5			99.46%
Pulrodemstat	KDM1/LSD1							98.86%
T-3775440 hydrochloride	KDM1/LSD1							99.13%
INCB059872	LSD1							99.60%
GSK 690 Hydrochloride	KDM1/LSD1							98.58%
GSK-J1 lithium salt						KDM6		98.33%
INCB059872 dihydrochloride	LSD1							99.64%
HDAC6-IN-3	KDM1/LSD1							98.0%
CBB1007 trihydrochloride	KDM1/LSD1, IC₅₀: 5.27 μM
NCGC00247743				KDM4				99.38%
LSD1-IN-30	LSD1, IC₅₀: 0.291 μM							99.03%
DDP-38003 trihydrochloride	KDM1/LSD1
KDM4-IN-2				KDM4				98.29%
NCDM-32B				KDM4A, IC₅₀: 3 μM KDM4C, IC₅₀: 1 μM
CBB1007 hydrochloride	KDM1/LSD1, IC₅₀: 5.27 μM							98.0%
CBB1007	KDM1/LSD1, IC₅₀: 5.27 μM
LSD1-IN-5	KDM1/LSD1
LSD1-IN-6	KDM1/LSD1
Pulrodemstat Methylbenzenesulfonate	KDM1/LSD1
T-448 free base	KDM1/LSD1
PROTAC KDM4 degrader-1				KDM4A, DC₅₀: 37.53 nM KDM4B, DC₅₀: 39.93 nM KDM4C, DC₅₀: 49.41 nM
LSD1/HDAC6-IN-1	KDM1/LSD1
LSD1-IN-13 hydrochloride	KDM1/LSD1
MC2652	KDM1/LSD1
MC4491	LSD1, IC₅₀: 0.152 μM
KDM4-IN-4				KDM4A-Tudor domain, Ki: 80 μM
LSD1-IN-31	LSD1
LSD1-IN-17	KDM1/LSD1
3β-Acetoxyl-atractylenolide I	LSD1, IC₅₀: 57 μM
LSD1-IN-34	LSD1, IC₅₀: 4.51 nM
XL177A (GMP)						KDM6
LSD1-IN-43	KDM1/LSD1
HSP90/LSD1-IN-1	LSD1
KDM4 ligand-1				KDM4A KDM4B KDM4C
LSD1-IN-15	KDM1/LSD1
NCD38	LSD1
LSD1-IN-49	LSD1, IC₅₀: 29 nM
DDP-38003	KDM1/LSD1, IC₅₀: 84 nM
LSD1-UM-109	LSD1, IC₅₀: 3.1 nM
LSD1-IN-41	LSD1
LSD1-IN-38	LSD1, IC₅₀: 1.2 nM
INCB059872 TFA	LSD1
KDM4C-IN-2				KDM4C, IC₅₀: 147 μM KDM4C, Ki: 51 μM
INCB059872 tosylate	LSD1
S1427	KDM1/LSD1
LSD1-IN-23	KDM1/LSD1, IC₅₀: 0.58 μM
LSD1/2-IN-4	KDM1/LSD1
NCL1	LSD1, IC₅₀: 2.5 ± 0.5 μM
cis-4-Br-2,5-F2-PCPA	KDM1/LSD1
KDM1/CDK1-IN-1	KDM1/LSD1
LSD1/HDAC-IN-2	KDM1/LSD1, IC₅₀: 39.0 nM
DW-229		KDM2	KDM3	KDM4A	KDM5B	KDM6
LSD1-IN-26	LSD1, IC₅₀: 25.3 ± 1.4 nM
LSD1-IN-21	LSD1, IC₅₀: 0.956 μM
KDM5-C49					KDM5
LSD1-IN-48	LSD1, IC₅₀: 7.87 nM
LSD1-IN-35	LSD1
LSD1-IN-18	KDM1/LSD1
N19-0881					KDM5
LSD1-IN-25	LSD1, IC₅₀: 46 nM LSD1, Ki: 30.3 nM
(1S,2R)-Tranylcypromine hydrochloride	KDM1/LSD1
YTHu78					KDM5B
LSD1-IN-46	LSD1, IC₅₀: 0.082 μM
TAS1440	KDM1/LSD1, IC₅₀: 4.8 nM
LSD1-IN-22	KDM1/LSD1
LSD1-IN-39	LSD1, IC₅₀: 0.18 μM
LSD1-IN-19	KDM1/LSD1
MC4455	LSD1
LSD1-IN-42	LSD1, IC₅₀: 0.08 μM
LSD1-IN-10	LSD1, IC₅₀: 5 nM
LSD1/2-IN-3	KDM1/LSD1
LSD1-IN-49 hydrochloride	LSD1, IC₅₀: 29 (hLSD1) nM
DC551040	LSD1, IC₅₀: 2.14 nM
LSD1-IN-16	KDM1/LSD1
LSD1-IN-45	LSD1
Pulrodemstat hydrochloride	KDM1/LSD1
Tranylcypromine-d₅ hydrochloride	KDM1/LSD1							99.42%
AW4	LSD1
LSD1/HDAC-IN-1	LSD1, IC₅₀: 0.571 μM
JQKD82					KDM5
LSD1/ER-IN-1	KDM1/LSD1
LSD1-IN-36	LSD1, IC₅₀: 0.8 nM
CBB1003 hydrochloride	KDM1/LSD1
EPZ020809				KDM4C, Ki: 31 nM
LSD1-IN-44	LSD1-CoREST, IC₅₀: 0.02 μM
MC3935	LSD1-CoREST, IC₅₀: 0.52 μM

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